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Constrained amino alcohols
SpiroKit 6: Constrained amino alcohols

Why SpiroKit 6?

The introduction of the very hydrophilic hydroxyl group can cause some metabolism-related troubles which can be circumvented by:

  • A constrained structure which will not fit active site or will not adopt transition state
  • The introduction of hindered groups to block conjugation reactions

To help medicinal chemists save time in their research programs, SpiroChem has selected a smart set of 54 constrained hindered amino alcohol derivatives.

SpiroKit 6: Constrained amino alcohols

Offered subsets

SPIROKIT 6a : Bridged amino alcohols

A selection of 6 bridged amino secondary alcohols.

Catalog ID Compounds Amount (each) Price (whole set)
SPK6a 6 100mg CHF 940 USD 1.090
250mg CHF 1.610 USD 1.790
500mg CHF 2.740 USD 2.990

A selection of 5 spiro and fused amino secondary alcohols.

Catalog ID Compounds Amount (each) Price (whole set)
SPK6b 5 100mg CHF 670 USD 730
250mg CHF 1.030 USD 1.130
500mg CHF 1.570 USD 1.730

A selection of 14 constrained amino alcohols (secondary amines) with OH shielding to prevent from conjugaison reactions.

Catalog ID Compounds Amount (each) Price (whole set)
SPK6c 14 100mg CHF 1.390 USD 1.530
250mg CHF 1.950 USD 2.130
500mg CHF 3.010 USD 3.290

A selection of 5 constrained amino alcohols (primary amines) with OH shielding to prevent from conjugation reactions.

Catalog ID Compounds Amount (each) Price (whole set)
SPK6d 5 100mg CHF 740 USD 820
250mg CHF 1.240 USD 1.390
500mg CHF 1.850 USD 2.030

A selection of 6 constrained amino alcohols (secondary amines) with OH shielding with a CF3 group.

Catalog ID Compounds Amount (each) Price (whole set)
SPK6e 6 100mg CHF 790 USD 890
250mg CHF 990 USD 1.090
500mg CHF 1.450 USD 1.590

A selection of 10 spiro Boc amino alcohols.

Catalog ID Compounds Amount (each) Price (whole set)
SPK6f 10 100mg CHF 1.590 USD 1.790
250mg CHF 2.490 USD 2.790
500mg CHF 3.750 USD 4.150

A selection of 8 fused and bridged Boc amino alcohols.

Catalog ID Compounds Amount (each) Price (whole set)
SPK6g 8 100mg CHF 1.350 USD 1.490
250mg CHF 2.210 USD 2.430
500mg CHF 3.290 USD 3.610
SpiroKit 6: Constrained amino alcohols

More Information

To receive more information about the SpiroKits, please contact Laurence Jung, PhD: laurence.jung@spirochem.com

SpiroKits

Other SpiroKits

SpiroKit 1

pKa-Tuned
Amines

SpiroKit 2

sp2 to sp3
Switch

SpiroKit 3

Constrained
Amino Acids

SpiroKit 4

Azaspiro[3.3]heptane derivatives

SpiroKit 5

Bicyclic diamines

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